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| DiscoveryProbe™ Epigenetics Compound Library
A unique collection of 240 epigenetics-related small molecules for epigenetics reasearch. |
Sample solution is provided at 25 µL, 10mM.
Click and Customize the Panel with your own choices of compounds/size/quantities/chemical forms etc.
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| Catalog No. | Product Name | Summary | Targets | CAS Number | Smiles | |
| A3692 | OTX-015 | BRD inhibitor | Bromodomain | 202590-98-5 | CC1=C(SC2=C1C(=NC(C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C | |
| A4093 | ITF2357 (Givinostat) | HDAC inhibitor | HDAC | 732302-99-7 | CCN(CC)CC1=CC2=C(C=C(COC(NC3=CC=C(C(NO)=O)C=C3)=O)C=C2)C=C1.O.Cl | |
| A4138 | Tofacitinib (CP-690550,Tasocitinib) | Janus kinase inhibitor | JAK | 477600-75-2 | CC1CCN(CC1N(C)C2=NC=NC3=C2C=CN3)C(=O)CC#N | |
| A4166 | EPZ5676 | DOT1L inhibitor,potent and SAM competitive | Histone Methyltransferase | 1380288-87-8 | CC(C)N(CC1C(C(C(O1)N2C=NC3=C2N=CN=C3N)O)O)C4CC(C4)CCC5=NC6=C(N5)C=C(C=C6)C(C)(C)C | |
| A8708 | Sephin1 | Selective PPP1R15A inhibitor | Protein Ser/Thr Phosphatases | 13098-73-2 | ClC1=CC=CC=C1/C=N/NC(N)=N | |
| A8712 | MCB-613 | stimulator of steroid receptor coactivator (SRC) | Histone Acetyltransferases | 1162656-22-5 | O=C(/C(CN(CC)C/1)=C/C2=CC=CN=C2)C1=C\C3=CN=CC=C3 | |
| B1499 | RVX-208 | Potent BET bromodomain inhibitor | Bromodomain | 1044870-39-4 | CC1=CC(=CC(=C1OCCO)C)C2=NC(=O)C3=C(C=C(C=C3N2)OC)OC | |
| B4891 | ML324 | JMJD2 demethylase inhibitor, potent and cell-permeable | Histone Demethylases | 1222800-79-4 | OC1=CC(C2=CC=C(C(NCCCN(C)C)=C)C=C2)=CC3=CC=CN=C31 | |
| Download the Epigenetics-Compound-Library - XLSX Download the Epigenetics-Compound-Library - SDF | ||||||
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| Form | Pre-dissolved DMSO solutions | Stability | -20°C: 12 months -80°C: 24 months |
| Packaging | 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode. | ||
| General tips | For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months. | ||
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
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Available in stock with overnight delivery and free shipping over $500
Cost-effective and competitive price to save your findings
Potent, selective and cell-permeable in inhibiting or activating target molecules
Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)
Detailed files describing potency, selectivity and applications etc.
Supported by published data from top peer-reviewed journals
Guaranteed high quality with NMR and HPLC validation
