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- A4022 BMS-708163 (Avagacestat)Summary: γ-secretase inhibitor
- A8621 Bestatin hydrochlorideTarget: AminopeptidasesSummary: Inhibitor of aminopeptidase N (APN)/CD13 and aminopeptidase B.
- B7535 Eeyarestatin ITarget: ERADSummary: inhibitor of endoplasmic reticulum-associated degradation (ERAD) and protein translocation
- B5306 Obestatin (rat)Summary: Endogenous peptide that suppresses food intake and body weight-gain
- B5332 CatestatinSummary: Non-competitive nicotinic cholinergic antagonist
- B6319 AlrestatinSummary: aldose reductase inhibitor
- B1037 AlvelestatTarget: NESummary: NE inhibitor
- A8190 Semagacestat (LY450139)Summary: γ-secretase inhibitor
- A4430 Sivelestat sodium saltTarget: ElastasesSummary: Leukocyte elastase inhibitor
- A4406 BegacestatSummary: γ-secretase inhibitor